Combining LY2880070 with Gemcitabine for treating Ewing Sarcoma and similar tumors

A Phase II Study of Oral CHK1 Inhibitor LY2880070 in Combination With Low-Dose Gemcitabine in Patients With Relapsed or Refractory Ewing Sarcoma, Ewing-like Sarcoma, and Desmoplastic Small Round Cell Tumor

Phase 2 Interventional Memorial Sloan Kettering Cancer Center · NCT05275426

This study is testing if combining a new drug called LY2880070 with the chemotherapy gemcitabine can help people with Ewing sarcoma or similar tumors get better results from their treatment.

Quick facts

PhasePhase 2
Study typeInterventional
Enrollment24 (estimated)
SexAll
SponsorMemorial Sloan Kettering Cancer Center Academic / other
Drugs / interventionschemotherapy, radiation, cyclophosphamide, doxorubicin
Locations1 site (New York, New York)
Trial IDNCT05275426 on ClinicalTrials.gov

What this trial studies

This study investigates the effectiveness of LY2880070 in combination with the chemotherapy drug gemcitabine for patients diagnosed with Ewing sarcoma or Ewing-like sarcoma. It aims to determine if this combination can improve treatment outcomes for patients with these specific types of cancer. The study will include patients with histologically confirmed locally advanced or metastatic disease, focusing on those with specific molecular characteristics. Participants must meet certain eligibility criteria, including weight and age requirements.

Who should consider this trial

Good fit: Ideal candidates for this study are patients with locally advanced or metastatic Ewing sarcoma or Ewing-like sarcoma who meet the specified molecular criteria.

Not a fit: Patients with other types of sarcomas or those who do not meet the molecular criteria for Ewing sarcoma or Ewing-like sarcoma may not benefit from this study.

Why it matters

Potential benefit: If successful, this treatment could provide a new effective option for patients suffering from Ewing sarcoma and related tumors.

How similar studies have performed: While this specific combination is being tested in this trial, similar approaches have shown promise in other studies targeting Ewing sarcoma and related conditions.

Eligibility criteria

Show full inclusion / exclusion criteria
Inclusion Criteria:

* Consent/Assent: all patients and/or their parents or legally authorized representatives must sign written informed consent; assent, when appropriate, will be obtained according to institutional guidelines
* Weight/Age: patients must be ≥40 kg at the time of study enrollment, but may be of any age
* Diagnosis: Patients must have histologically documented locally advanced or metastatic disease confirmed at MSK as follows:

  * Main cohort: Ewing sarcoma as molecularly defined by an EWSR1 fusion with an ETS-transcription factor family member including FLI1, ERG, ETV1, ETV4, and FEV
  * Pilot cohort: Ewing-like sarcomas including CIC-rearranged sarcoma, BCOR-rearranged sarcoma, and sarcomas with a rearrangement between EWSR1 and a non-ETS family gene or desmoplastic small round cell tumor as molecularly defined by an EWSR1-WT1 fusion

Note: Any patient being enrolled into the pilot cohort that does not have a CIC, BCOR- rearranged sarcoma, or desmoplastic small round cell tumor will be reviewed with study pathologist, Dr. Cristina Antonescu, to ensure the categorization as Ewing-like sarcoma is appropriate

* Patients must be able to swallow capsules
* Therapeutic options: patient's current disease state must be one which has failed standard cytotoxic chemotherapy including cyclophosphamide/doxorubicin/vincristine and ifosfamide/etoposide
* Disease Status: patients must have measurable disease based on RECIST 1.1
* Performance level: Karnofsky ≥70% for patients \>16 years of age and Lansky ≥70 for patients ≤16 years of age
* Prior Therapy: patients may have had any number of regimens and must meet the following minimum duration from prior anti-cancer directed therapy prior to enrollment

Note: Patients who have previously received gemcitabine will be allowed unless they had hypersensitivity or unacceptable toxicity attributed to gemcitabine

* ≥ 21 days must have elapsed after the last dose of cytotoxic or myelosuppressive chemotherapy and patients must have recovered from the acute toxic effects of these agents (other than alopecia)
* ≥ 14 days must have elapsed after radiation therapy, and toxicity related to prior radiation therapy must be recovered to grade ≤ 1
* ≥ 21 days must have elapsed after the last dose of antibody therapy, and toxicity related to prior antibody therapy must be recovered to grade ≤ 1

Organ Function Requirements:

* Adequate bone marrow function defined as:

  * Absolute neutrophil count (ANC) ≥ 1500/mm3
  * Platelet count ≥ 100,000/mm3
  * Hemoglobin ≥ 8 g/dl
* Adequate renal function defined as estimated glomerular filtration (eGFR) rate ≥ 60 mL/min/1.73m2:

  * as estimated by CKD-EPI equation for patients ≥ 18 years of age OR
  * As estimated by cystatin C for patients \< 18 years of age
* Adequate liver function defined as:

  * Bilirubin (sum of conjugated + unconjugated) ≤ 1.5 x upper limit of normal for age
  * AST or ALT ≤ 2.5 x upper limit of normal for patients without liver metastases
  * AST or ALT ≤ 5 x upper limit of normal for patients with liver metastases
  * Serum albumin ≥ 2.5 g/dl
* Adequate cardiac function defined as:

  * Left ventricular ejection fraction (LVEF) \>45% as measured on echocardiogram, cardiac MRI, or MUGA
  * QTc \< 470 ms on screening 12 lead electrocardiogram
* Pregnancy/Contraception

  * Post-menarchal females must have a negative urine or serum pregnancy test at screening and ≤ 24 hours prior to study treatment
  * Males or females of reproductive potential must be willing to use a barrier method of contraception throughout the course of the study and for 6 months after completing study treatment

Exclusion Criteria:

* Patients for whom the investigator deems that gemcitabine is not appropriate
* Patients who have an uncontrolled infection
* Central Nervous System (CNS) Metastases

  * Patients who have symptomatic central nervous system (CNS) metastases. Note: patients with treated and asymptomatic CNS metastases are eligible.
  * Patients with CNS metastases requiring corticosteroids for management
  * If the treatment of CNS disease requires anticonvulsants, the dose must have been stable for ≥ 4 weeks.
* Patients who are pregnant or breast feeding
* Patients who have a history of Torsades de Pointes, carry a diagnosis of congestive heart failure, or have a family history of prolonged QT syndrome
* Patients who, in the opinion of the investigator, may not be able to comply with the safety monitoring requirements of the study
* Patients with known hypersensitivity to gemcitabine

Where this trial is running

New York, New York

Study contacts

How to participate

  1. Review the eligibility criteria above with your treating physician.
  2. Visit the official trial page on ClinicalTrials.gov for the most current contact information and recruitment status.
  3. Contact the listed study coordinator or principal investigator to request pre-screening. Pre-screening is free and never obligates you to enroll.
Conditions Ewing SarcomaEwing-Like SarcomaLY2880070Gemcitabine21-428Memorial Sloan Kettering Cancer Center
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.