Using targeted therapy to treat hereditary colorectal cancer by focusing on DNA mismatches

Targeting DNA Mismatches for Auger Electron Radiotherapy

NIH-funded research Hunter College · NIH-10751210

This study is exploring a new way to treat hereditary colorectal cancer by using a special technology that targets and fixes mistakes in DNA that can cause tumors, which might make radiation therapy work better for patients with this condition.

Quick facts

Grant typeR21 grant
Study typeNIH-funded research
Funding institutionHunter College NIH-funded
Lab location1 site (New York, United States)
Project IDNIH-10751210 on NIH RePORTER

What this research studies

This research investigates a novel approach to treating hereditary colorectal cancer by targeting mismatched DNA base pairs that can lead to tumor development. The study utilizes a technology called metalloinsertors, which bind specifically to these mismatches and disrupt their formation, potentially enhancing the effectiveness of radiotherapy. By employing iodine-123, an Auger electron-emitting radionuclide, the research aims to develop a targeted radiotherapeutic that could selectively destroy cancer cells with DNA repair deficiencies. Patients with hereditary non-polyposis colorectal cancer may benefit from this innovative treatment strategy.

Who could benefit from this research

Good fit: Ideal candidates for this research are individuals diagnosed with hereditary non-polyposis colorectal cancer or those with known mismatch repair deficiencies.

Not a fit: Patients without hereditary colorectal cancer or those whose cancer is not associated with DNA mismatch repair deficiencies may not benefit from this research.

Why it matters

Potential benefit: If successful, this research could provide a new targeted treatment option for patients with hereditary colorectal cancer, improving their outcomes.

How similar studies have performed: While the approach of using metalloinsertors is relatively novel, previous research has shown promise in targeting DNA mismatches for therapeutic purposes.

Where this research is happening

New York, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Hereditary Non-Polyposis Colon CancerHereditary Nonpolyposis Colo-rectal CancerHereditary Nonpolyposis Colon CancerHereditary Nonpolyposis Colorectal CancerLynch Syndrome
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.