New treatment for advanced prostate cancer using a novel therapeutic probe

A Dosimetry Study and Dose-escalation and of [177Lu]Lu-LNC1011 in Metastatic Castration-Resistant Prostate Cancer Patients

PHASE1; PHASE2 · Peking Union Medical College Hospital · NCT06250244

This study is testing a new treatment for advanced prostate cancer to see if it is safe and effective for patients whose cancer has spread and is resistant to other therapies.

Quick facts

PhasePHASE1; PHASE2
Study typeInterventional
Enrollment12 (estimated)
Ages18 Years to 80 Years
SexMale
SponsorPeking Union Medical College Hospital (other)
Locations1 site (Beijing, Beijing)
Trial IDNCT06250244 on ClinicalTrials.gov

What this trial studies

This clinical trial investigates the safety and efficacy of 177Lu-LNC1011, a new long-circulating PSMA therapeutic probe, in patients with metastatic castration-resistant prostate cancer (mCRPC). The study employs an open-label, non-randomized design with a 3+3 dose-escalation approach, starting treatment at a dose of 1.85 GBq over six weeks and escalating doses by 50% until dose-limiting toxicity is observed. The primary goals are to determine the maximum tolerated dose, assess safety, and evaluate initial treatment efficacy in this patient population.

Who should consider this trial

Good fit: Ideal candidates for this study are men with progressive metastatic castration-resistant prostate cancer and confirmed high PSMA expression.

Not a fit: Patients with significant renal impairment, low blood counts, or other serious health conditions may not benefit from this study.

Why it matters

Potential benefit: If successful, this treatment could provide a new therapeutic option for patients with advanced prostate cancer that is resistant to standard hormone therapies.

How similar studies have performed: While this approach is novel, similar studies targeting PSMA in prostate cancer have shown promising results, indicating potential for success.

Eligibility criteria

Show full inclusion / exclusion criteria
Inclusion Criteria:

* progressive metastatic castration-resistant prostate cancer
* tumors with high PSMA expression confirmed on 68Ga-PSMA PET/CT PSMA expression confirmed on 68Ga-PSMA PET/CT

Exclusion Criteria:

* a serum creatinine level of more than 150 μmol per liter
* a hemoglobin level of less than 10.0 g/dl
* a white-cell count of less than 4.0× 109/L
* a platelet count of less than 100 × 109/L
* a total bilirubin level of more than 3 times the upper limit of the normal range
* a serum albumin level of more than 3.0 g per deciliter
* cardiac insufficiency

Where this trial is running

Beijing, Beijing

Study contacts

How to participate

  1. Review the eligibility criteria above with your treating physician.
  2. Visit the official trial page on ClinicalTrials.gov for the most current contact information and recruitment status.
  3. Contact the listed study coordinator or principal investigator to request pre-screening. Pre-screening is free and never obligates you to enroll.

View on ClinicalTrials.gov →

Conditions: Metastatic Castration-resistant Prostate Cancer, PSMA, 177Lu, mCRPC

Last reviewed 2026-05-15 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.