Why some advanced prostate cancers stop responding to AR-blocking drugs

Identify Mechanisms Driving Resistance to AR Antagonists in CRPC

NIH-funded research Beth Israel Deaconess Medical Center · NIH-11198067

This research looks at why advanced prostate cancer keeps growing despite AR-blocking medicines like enzalutamide, to help men with castration-resistant prostate cancer.

Quick facts

Grant typeP01 program project
Study typeNIH-funded research
Funding institutionBeth Israel Deaconess Medical Center NIH-funded
Lab location1 site (Boston, United States)
Project IDNIH-11198067 on NIH RePORTER

What this research studies

The team grows prostate cancer cells in the lab that became resistant to AR antagonists and studies the changes that let the androgen receptor keep working, with a focus on a common truncated form called AR‑V7. They use genetic tools (including CRISPR-based methods), chromatin accessibility and DNA-binding analyses, and compare lab findings to tumor samples to link results to real patients. By mapping where AR and cooperating factors bind DNA and how chromatin is remodeled, they aim to reveal molecular targets for new tests or treatments.

Who could benefit from this research

Good fit: Men with castration-resistant prostate cancer, especially those whose disease progressed while on AR antagonists such as enzalutamide, are the most relevant group for this research.

Not a fit: People without prostate cancer or those whose tumors no longer rely on the androgen receptor are unlikely to benefit directly from this project.

Why it matters

Potential benefit: If successful, this work could lead to tests that predict resistance and new treatments that help men whose cancers stop responding to AR antagonists.

How similar studies have performed: Previous studies have linked AR‑V7 and chromatin changes to drug resistance, so this project builds on established findings but translating those insights into effective treatments remains experimental.

Where this research is happening

Boston, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.