Understanding a Protein Called SETDB1 in Lung Cancer

Dissecting the Mechanism of SETDB1 and its K867 Monoubiquitination in Lung Cancer Progression

NIH-funded research Roswell Park Cancer Institute Corp · NIH-11141731

This research explores how a protein named SETDB1 contributes to lung cancer growth, especially in patients with certain genetic changes, to find new ways to treat the disease.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionRoswell Park Cancer Institute Corp NIH-funded
Lab location1 site (Buffalo, United States)
Project IDNIH-11141731 on NIH RePORTER

What this research studies

Non-small cell lung cancer (NSCLC) is a serious illness, and while some targeted treatments exist, options for tumors with common KRAS mutations are still limited. This project focuses on a protein called SETDB1, which is often found in higher amounts in many cancers, including NSCLC, and seems to help tumors grow. We want to understand exactly how SETDB1 works in lung cancer cells and how a specific modification to it, called K867 monoubiquitination, affects its function. By uncovering these details, we hope to identify new weaknesses in lung cancer that could lead to more effective treatments, particularly for those with KRAS mutations.

Who could benefit from this research

Good fit: This foundational research is for patients with non-small cell lung cancer, particularly those with KRAS mutations, who may benefit from future targeted therapies developed from these findings.

Not a fit: Patients without non-small cell lung cancer or those whose cancer does not involve the specific mechanisms being studied may not directly benefit from this particular research.

Why it matters

Potential benefit: If successful, this research could lead to the discovery of new drug targets and treatment strategies for non-small cell lung cancer, especially for patients whose tumors have KRAS mutations.

How similar studies have performed: While targeted therapies for other lung cancer mutations have shown success, understanding the specific role of SETDB1 and its modifications in KRAS mutant NSCLC represents a novel and less explored area.

Where this research is happening

Buffalo, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.