Targeting tiny genetic switches in gene messages to treat inherited diseases

Identifying regulatory uORFs as a targetable axis for hereditary disease

NIH-funded research University of Pennsylvania · NIH-11113825

This project tests whether small sequences at the front of gene messages can be changed to raise or lower protein levels for people with inherited disorders.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of Pennsylvania NIH-funded
Lab location1 site (Philadelphia, United States)
Project IDNIH-11113825 on NIH RePORTER

What this research studies

Researchers will search large human genetic databases (like gnomAD, the Penn Medicine BioBank, and the UK Biobank) to find short regulatory sequences called upstream open reading frames (uORFs) that affect how much protein a gene makes. They will build a searchable, public database of these uORFs and use computer models to rank the most promising targets. Laboratory experiments using cell-based luciferase assays will check whether altering those uORFs actually changes protein output. The team will iterate between the computer predictions and lab results to refine which uORFs are best suited for future therapies.

Who could benefit from this research

Good fit: People with inherited conditions caused by abnormal protein levels—such as disorders linked to specific genes like BMPR2—would be the most relevant group for this research.

Not a fit: Patients with non-genetic problems (for example infections, injuries, or conditions not driven by gene expression changes) are unlikely to benefit directly from this work.

Why it matters

Potential benefit: If successful, this work could uncover new drug targets that let doctors increase or decrease specific proteins to treat some hereditary diseases.

How similar studies have performed: Laboratory studies have shown uORFs can control protein production, but using them broadly as therapeutic targets is a relatively new and largely unproven strategy in patients.

Where this research is happening

Philadelphia, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.