Targeting a specific variant of the androgen receptor in advanced prostate cancer

Targeting AR variants in advanced prostate cancer

NIH-funded research University of California at Davis · NIH-10538636

This study is looking at new ways to help men with advanced prostate cancer that doesn't respond to common treatments by targeting a specific part of the cancer called AR-V7, with the hope of making existing therapies work better.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of California at Davis NIH-funded
Lab location1 site (Davis, United States)
Project IDNIH-10538636 on NIH RePORTER

What this research studies

This research focuses on advanced prostate cancer that has become resistant to standard treatments like enzalutamide and abiraterone. It investigates the role of a specific variant of the androgen receptor, known as AR-V7, which contributes to this resistance. The researchers are developing new small molecule inhibitors that specifically target AR-V7 to improve treatment outcomes. By synthesizing and testing these novel compounds, they aim to enhance the effectiveness of existing therapies for patients with castration-resistant prostate cancer.

Who could benefit from this research

Good fit: Ideal candidates for this research are men diagnosed with castration-resistant prostate cancer who have not responded to standard anti-androgen therapies.

Not a fit: Patients with early-stage prostate cancer or those who have not yet undergone treatment with enzalutamide or abiraterone may not benefit from this research.

Why it matters

Potential benefit: If successful, this research could provide a new treatment option for patients with advanced prostate cancer who have developed resistance to current therapies.

How similar studies have performed: While targeting AR-V7 is a novel approach, previous studies have shown promise in targeting androgen receptor variants in cancer treatment, indicating potential for success.

Where this research is happening

Davis, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Anti-Cancer Agents
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.