Targeting a specific enzyme to treat breast cancer that has spread to the brain

Targeting FASN to eliminate metastatic breast cancer in the brain

NIH-funded research University of Toledo Health Sci Campus · NIH-10884918

This study is looking at how a common enzyme in breast cancer that spreads to the brain can be targeted using everyday heartburn medications to make cancer treatments work better for patients.

Quick facts

Grant typeR21 grant
Study typeNIH-funded research
Funding institutionUniversity of Toledo Health Sci Campus NIH-funded
Lab location1 site (Toledo, United States)
Project IDNIH-10884918 on NIH RePORTER

What this research studies

This research focuses on addressing metastatic breast cancer in the brain, a challenging condition due to the protective blood-brain barrier. The study investigates the role of fatty acid synthase (FASN), an enzyme that is found to be elevated in breast cancer brain metastasis. By repurposing FDA-approved proton pump inhibitors (PPIs), the research aims to inhibit FASN activity and enhance the effectiveness of existing cancer treatments. Patients may benefit from a novel approach that combines these inhibitors with standard therapies to improve outcomes.

Who could benefit from this research

Good fit: Ideal candidates for this research are breast cancer patients who have developed metastasis in the brain, particularly those with triple-negative breast cancer.

Not a fit: Patients with breast cancer that has not metastasized to the brain or those with other types of cancer may not benefit from this research.

Why it matters

Potential benefit: If successful, this research could provide a new treatment option for breast cancer patients with brain metastasis, potentially improving survival rates and quality of life.

How similar studies have performed: Previous studies have shown promise in targeting FASN with repurposed drugs, indicating potential for success in this novel approach.

Where this research is happening

Toledo, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.