Tabernanthalog for opioid addiction

Target Specificity of Tabernanthalog Treatment in Opioid Use Disorder

NIH-funded research University of Alabama at Birmingham · NIH-11363767

This project looks at whether tabernanthalog can help people with opioid use disorder by restoring prefrontal brain connections and lowering relapse risk.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of Alabama at Birmingham NIH-funded
Lab location1 site (Birmingham, United States)
Project IDNIH-11363767 on NIH RePORTER

What this research studies

Researchers are studying tabernanthalog, a compound related to psychedelics but designed to avoid hallucinations, to see if it can promote healthy brain wiring in the prefrontal cortex that helps control cravings. They will use laboratory and preclinical models to measure changes in neural connections and behaviors linked to opioid seeking and relapse, and will probe how the drug interacts with serotonin receptors. The team will investigate receptor specificity to reduce potential side effects such as cardiac or sensory disturbances. Successful preclinical results would support moving toward early human trials to test safety and benefit.

Who could benefit from this research

Good fit: People with opioid use disorder, especially those with repeated relapse or poor response to current medications, would be the likely candidates for future trials.

Not a fit: People without opioid use disorder or those seeking an already approved immediate treatment are unlikely to receive direct benefit from this research at its current preclinical stage.

Why it matters

Potential benefit: If successful, this work could lead to treatments that restore decision-making circuits, reduce relapse, and lessen the need for long-term opioid-substitution medications.

How similar studies have performed: Psychedelic drugs and ibogaine analogs have shown anti-addiction effects in animal models and some early human reports, but tabernanthalog is a newer non-hallucinogenic candidate with primarily preclinical evidence so far.

Where this research is happening

Birmingham, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.