Protease-blocking medicines for COVID-19

SARS-CoV-2 protease inhibitors for treating COVID-19

NIH-funded research Purdue University · NIH-10848439

Developing new medicines that block key coronavirus enzymes to help people with COVID-19.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionPurdue University NIH-funded
Lab location1 site (West Lafayette, United States)
Project IDNIH-10848439 on NIH RePORTER

What this research studies

Researchers at Purdue are designing and testing small-molecule drugs that block two viral enzymes (3CLpro and PLpro) SARS-CoV-2 needs to replicate. They will build on prior antiviral chemistry that worked against SARS and MERS, using lab binding and activity assays, bioavailability testing, and animal models to find the most promising compounds. The team aims to optimize safety and how the drugs behave in the body before moving lead candidates toward clinical testing. If a candidate looks good in preclinical work, it could advance into human trials at Purdue and collaborating sites.

Who could benefit from this research

Good fit: Once human trials begin, ideal participants would be people with confirmed SARS-CoV-2 infection, especially those early in illness or at higher risk of severe disease.

Not a fit: People without an active COVID-19 infection or those whose illness is driven mainly by late immune damage rather than viral replication are unlikely to benefit from antiviral protease inhibitors.

Why it matters

Potential benefit: If successful, these drugs could shorten or prevent severe COVID-19 by stopping the virus from multiplying in the body.

How similar studies have performed: Related protease inhibitors (for example drugs targeting the same viral protease) have shown clinical benefit, and this work builds on earlier successful antiviral chemistry for SARS and MERS.

Where this research is happening

West Lafayette, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-09 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.