Preventing resistance to KRAS-targeted treatments in colorectal cancer

Overcoming adaptive feedback resistance to KRAS inhibition in colorectal cancer

NIH-funded research Massachusetts General Hospital · NIH-11306623

Researchers are combining drugs to help people with KRAS-mutant colorectal cancer respond better and longer to new KRAS-targeted therapies.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionMassachusetts General Hospital NIH-funded
Lab location1 site (Boston, United States)
Project IDNIH-11306623 on NIH RePORTER

What this research studies

At Massachusetts General Hospital, the team is studying why colorectal tumors rapidly reactivate the KRAS pathway and stop KRAS inhibitors from working. They analyze tumor samples and lab models to map the adaptive feedback signals that drive resistance. The researchers test combinations of drugs (for example adding EGFR-targeting agents) in cell and preclinical models to find strategies that block pathway reactivation. Promising combinations will be prioritized to inform future clinical trials for patients.

Who could benefit from this research

Good fit: Ideal candidates are people with colorectal cancer whose tumors have KRAS mutations (such as G12C or G12D) and who are candidates for KRAS-targeted therapies or future combination trials.

Not a fit: Patients without KRAS-mutant tumors or whose cancers rely on different resistance pathways may not benefit from these specific combination approaches.

Why it matters

Potential benefit: Could lead to combination treatments that make KRAS-targeted drugs more effective and durable for colorectal cancer patients.

How similar studies have performed: Previous work showed combination approaches (for example adding EGFR blockade) improved outcomes in BRAF-mutant colorectal cancer, and KRASG12C inhibitors have strong responses in lung cancer but limited and less durable responses so far in colorectal cancer, so this approach has supportive precedent but remains unproven for KRAS-mutant CRC.

Where this research is happening

Boston, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Cancer ModelCancerModelCancers
Last reviewed 2026-06-10 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.