Methotrexate and other medicines for rhodopsin-related retinitis pigmentosa

Pharmacological studies of RHO-associated retinitis pigmentosa

NIH-funded research University of Pittsburgh at Pittsburgh · NIH-11295659

This project tests whether methotrexate and similar repurposed drugs can protect vision in people with rhodopsin-linked autosomal dominant retinitis pigmentosa.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of Pittsburgh at Pittsburgh NIH-funded
Lab location1 site (Pittsburgh, United States)
Project IDNIH-11295659 on NIH RePORTER

What this research studies

The team is focusing on repurposing methotrexate, a drug already used for cancer and rheumatoid arthritis, as a treatment for RHO-adRP. They will study how methotrexate acts on AMPK and adenosine signaling pathways, compare drug levels in the eye after different delivery routes, and use retinal explant assays to screen other approved drugs that might help. The work builds on preclinical studies and a recent clinical trial that reported improved retinal function after intravitreal methotrexate. The goal is to find safer long-term dosing and additional repurposed medicines that could slow or stop vision loss.

Who could benefit from this research

Good fit: People with genetically confirmed rhodopsin-associated autosomal dominant retinitis pigmentosa, especially those with progressive vision loss, would be the ideal candidates for related clinical work.

Not a fit: People with other genetic causes of retinal degeneration, those with very advanced retinal scarring that cannot be rescued, or those who cannot safely receive methotrexate may not benefit from these interventions.

Why it matters

Potential benefit: If successful, this work could produce a safe, long-term medicine or delivery approach that slows or prevents vision loss in people with RHO-associated adRP.

How similar studies have performed: Early laboratory studies and a recent small clinical trial reported that intravitreal methotrexate improved retinal function, but larger confirmatory trials are still needed.

Where this research is happening

Pittsburgh, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.