Improving radiation response in rectal cancer by targeting low-oxygen tumor areas

Tumor-Selective Radiosensitization by Targeting Hypoxia in Rectal Cancer

NIH-funded research Beckman Research Institute/city of Hope · NIH-11267984

Using an approved drug that lowers tumor oxygen use alongside radiation to help shrink rectal tumors in people with locally advanced rectal cancer.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionBeckman Research Institute/city of Hope NIH-funded
Lab location1 site (Duarte, United States)
Project IDNIH-11267984 on NIH RePORTER

What this research studies

If you have locally advanced rectal cancer and are getting pre-surgery chemotherapy and radiation (total neoadjuvant therapy), this project looks at adding a drug that reduces tumor oxygen use to make radiation more effective. Tumor areas with low oxygen (hypoxia) can resist radiation, and the team will give the FDA-approved drug papaverine during radiation to block tumor mitochondrial oxygen consumption and try to sensitize tumors. Researchers will follow response with imaging, endoscopy, and tissue samples and will study tumor biology to see who benefits and why. The aim is to increase complete responses so more people might avoid major surgery and its long-term consequences.

Who could benefit from this research

Good fit: Adults with locally advanced rectal adenocarcinoma who are scheduled for total neoadjuvant therapy (preoperative chemotherapy and radiation) are the ideal candidates.

Not a fit: Patients with early-stage disease, widespread metastatic cancer, or those unable to tolerate the study drug or radiation are unlikely to benefit from this approach.

Why it matters

Potential benefit: If successful, more patients could have their tumors fully controlled before surgery and avoid major rectal surgery and its lasting side effects.

How similar studies have performed: Preclinical data support that blocking mitochondrial oxygen use (for example with papaverine) can sensitize tumors to radiation, but translating this approach to rectal cancer patients is largely new.

Where this research is happening

Duarte, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
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Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.