How genes and blood metabolites affect HIV drug levels

Quantifying genomic and pharmacometabolomic differences in antiretroviral exposure in MACS/WIHS Combined Cohort Study

NIH-funded research University of California, San Francisco · NIH-11136554

This project uses blood samples and genetic data to connect people's genes and small molecules in the blood with levels of HIV medicines (dolutegravir and tenofovir) to better understand side effects and responses.

Quick facts

Grant typeR21 grant
Study typeNIH-funded research
Funding institutionUniversity of California, San Francisco NIH-funded
Lab location1 site (San Francisco, United States)
Project IDNIH-11136554 on NIH RePORTER

What this research studies

You would be part of research using time-series blood samples from the MACS/WIHS Combined Cohort Study to measure levels of dolutegravir (DTG) and tenofovir (from TAF) alongside the plasma metabolome and genetic markers. The team will compare how metabolite patterns and genetic differences link to drug concentrations in blood and cells and to metabolic side effects like weight gain and insulin resistance. This work focuses on diverse men and women, including groups often understudied, using intensive pharmacokinetic sampling already collected in the cohort. The goal is to find biomarkers that predict who has higher drug exposure or is at risk for metabolic adverse effects.

Who could benefit from this research

Good fit: Ideal candidates are people living with HIV who are taking dolutegravir or tenofovir (TAF) and who participate in or can provide samples to the MACS/WIHS Combined Cohort Study.

Not a fit: People who are not on these specific HIV medications or who cannot provide blood samples will be unlikely to benefit directly from this research.

Why it matters

Potential benefit: If successful, this could help personalize HIV treatment by identifying who is likely to have higher drug exposure or metabolic side effects so doctors can tailor therapies.

How similar studies have performed: Related pharmacometabolomic studies have predicted responses to drugs like sertraline, escitalopram, and aspirin, but applying these methods to HIV antiretrovirals is relatively new.

Where this research is happening

San Francisco, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Acquired Immune Deficiency Syndrome VirusAcquired Immunodeficiency Syndrome Virus
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.