FAP-targeted radioactive therapy that gets trapped inside pancreatic tumors

Lysosome Trapped FAP-Targeted Theranostics for Pancreatic Cancer

NIH-funded research University of Nebraska Medical Center · NIH-11286819

A radioactive medicine aimed at fibroblast-rich pancreatic tumors that stays inside cancer tissue to deliver stronger, more focused radiation for people with pancreatic cancer.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of Nebraska Medical Center NIH-funded
Lab location1 site (Omaha, United States)
Project IDNIH-11286819 on NIH RePORTER

What this research studies

Researchers are developing radioactive drugs that home to a protein called fibroblast activation protein (FAP), which is common in many pancreatic tumors. They are adding a lysosome-trapping chemical trick so the drug forms a bond inside tumor cells and remains in the tumor longer, using radioactive isotopes 177Lu and 225Ac to deliver radiation. The team will optimize how these compounds behave in tumors and normal tissues, study how pancreatic cancer biology affects trapping, and measure biodistribution and tumor retention. Although much of the work is preclinical, the aim is to create treatments that could later move into patient trials.

Who could benefit from this research

Good fit: Ideal candidates would be people with pancreatic ductal adenocarcinoma, especially those whose tumors show high fibroblast activation protein (FAP) expression or who have metastatic disease not controlled by standard therapies.

Not a fit: Patients without FAP-expressing tumors, with other cancer types, or who cannot receive radionuclide therapy would likely not benefit from this work.

Why it matters

Potential benefit: If successful, this approach could deliver higher doses of targeted radiation to pancreatic tumors while sparing normal tissues, potentially improving tumor control and reducing side effects.

How similar studies have performed: FAP-targeted imaging agents have successfully located tumors, but FAP-directed therapeutic radioligands have historically suffered from poor tumor retention, and the lysosomal trapping approach is a newer preclinical strategy with encouraging but unproven results.

Where this research is happening

Omaha, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Cancer CauseCancer EtiologyCancers
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.