DNA 'untangling' enzymes and their role in cancer

Understanding and exploiting DNA topoisomerases in cancer biology

NIH-funded research Johns Hopkins University · NIH-11175521

Researchers are learning how enzymes that untangle DNA affect cancer cells and cancer drugs, with the goal of improving treatments for people with cancer.

Quick facts

Grant typeNIH-funded research
Study typeNIH-funded research
Funding institutionJohns Hopkins University NIH-funded
Lab location1 site (Baltimore, United States)
Project IDNIH-11175521 on NIH RePORTER

What this research studies

If you or a loved one has cancer, this project focuses on enzymes called topoisomerase II that control DNA winding and untangling in cancer cells. The team will use biochemical experiments, structural imaging, computer modeling, and cell-based tests to see how these enzymes work, where they act on chromosomes, and how cancer drugs interact with them. They will also study how cellular metabolism (the TCA cycle) changes enzyme activity and how mistakes by the enzyme can cause DNA damage. The work is lab-based and aims to reveal mechanisms that could guide safer or more effective therapies in the future.

Who could benefit from this research

Good fit: People with cancers commonly treated with topoisomerase II–targeting drugs (for example certain leukemias, lymphomas, and breast cancers) or patients willing to donate tumor or blood samples for research would be most relevant.

Not a fit: Patients with cancers unrelated to topoisomerase II activity or those seeking immediate new treatment options are unlikely to receive direct benefit from this lab-focused research.

Why it matters

Potential benefit: If successful, this work could lead to better-targeted cancer drugs or strategies that reduce DNA damage from treatment.

How similar studies have performed: Drugs that target topoisomerase II (such as etoposide and doxorubicin) are already used in cancer care, so this work builds on established clinical approaches while addressing new mechanistic questions.

Where this research is happening

Baltimore, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Anti-Cancer AgentsCancer BiologyCancer CauseCancer DrugCancer Etiology
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.