Delta opioid receptors and migraine-related head pain

The role of delta opioid receptors in trigeminovascular pain

['FUNDING_R01'] · WASHINGTON UNIVERSITY · NIH-11322044

This work looks at whether medicines that activate delta opioid receptors can reduce severe migraine and medication-overuse headaches.

Quick facts

Phase['FUNDING_R01']
Study typeNih_funding
SexAll
SponsorWASHINGTON UNIVERSITY (nih funded)
Locations1 site (SAINT LOUIS, UNITED STATES)
Trial IDNIH-11322044 on ClinicalTrials.gov

What this research studies

Researchers are studying how activating delta opioid receptors affects head pain using laboratory models of medication-overuse headache and chronic migraine. They tested delta opioid receptor activators in animal headache models and found these drugs reversed medication-induced head pain in prior work. The team performed a large peptidomic screen and identified the PACAP/PAC1 system as a possible link between chronic migraine and medication overuse. They are mapping where delta opioid receptors and PACAP/PAC1 appear together in pain-processing regions to guide development of targeted therapies.

Who could benefit from this research

Good fit: People with chronic migraine who have developed medication-overuse headache from frequent use of acute headache drugs would be the most relevant group.

Not a fit: Patients whose headaches are not related to medication overuse or who have non-trigeminal headache disorders are less likely to benefit from these findings.

Why it matters

Potential benefit: If successful, this work could lead to new targeted medicines that relieve medication-overuse headache and improve quality of life without forcing patients to permanently stop helpful medications.

How similar studies have performed: Preclinical work from this team showed delta opioid receptor activators reversed medication-induced head pain in animal models, though human clinical evidence is still limited.

Where this research is happening

SAINT LOUIS, UNITED STATES

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.

View on NIH RePORTER →

Last reviewed 2026-05-15 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.