Creating a new targeted treatment for prostate cancer

Development of an Innovative PSMA-Targeted Small Molecule Prodrug for Prostate Cancer

NIH-funded research Cancer Targeted Technology, LLC · NIH-10910547

This study is testing a new treatment for advanced prostate cancer that aims to deliver a powerful cancer-fighting drug directly to the cancer cells, which could help improve results and lessen side effects for patients.

Quick facts

Grant typeSbir 2 grant
Study typeNIH-funded research
Funding institutionCancer Targeted Technology, LLC NIH-funded
Lab location1 site (Woodinville, United States)
Project IDNIH-10910547 on NIH RePORTER

What this research studies

This research focuses on developing a novel small molecule prodrug that targets prostate-specific membrane antigen (PSMA) to treat metastatic castration-resistant prostate cancer (mCRPC). The approach involves conjugating a potent cancer-fighting agent, monomethyl auristatin E (MMAE), to a targeting molecule that specifically binds to cancer cells, minimizing damage to healthy cells. By enhancing the delivery of the drug directly to the cancer cells, this method aims to improve treatment efficacy while reducing side effects. Patients may have the opportunity to participate in clinical trials evaluating this innovative treatment.

Who could benefit from this research

Good fit: Ideal candidates for this research are men diagnosed with metastatic castration-resistant prostate cancer who have limited treatment options.

Not a fit: Patients with early-stage prostate cancer or those who do not express the PSMA biomarker may not benefit from this research.

Why it matters

Potential benefit: If successful, this research could provide a more effective and less toxic treatment option for patients with advanced prostate cancer.

How similar studies have performed: While there have been successful applications of antibody-drug conjugates in other cancers, this specific approach using small molecule drug conjugates for mCRPC is relatively novel.

Where this research is happening

Woodinville, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-14 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.