CD4-like drugs that expose and disable HIV's outer coat so antibodies can kill infected cells

Probing functional HIV-1 envelope glycoprotein conformations with novel potent CD4-mimetic compounds

NIH-funded research Dana-Farber Cancer Inst · NIH-11113854

Small CD4-mimic molecules are being made to force open HIV’s outer protein so antibodies can better find and destroy infected cells, potentially helping people with HIV.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionDana-Farber Cancer Inst NIH-funded
Lab location1 site (Boston, United States)
Project IDNIH-11113854 on NIH RePORTER

What this research studies

If you have HIV, this project is creating tiny molecules that latch onto the virus’s envelope protein and make it change shape. Those changes block the virus from entering cells and reveal hidden sites that antibodies can bind. The team will design and test different CD4-mimetic compounds in the lab and in animal models to find the most potent ones. Promising compounds will be studied for how well they work together with antibodies to reduce infected cells or prevent infection.

Who could benefit from this research

Good fit: Ideal future participants would be people living with HIV, particularly those on suppressive antiretroviral therapy who still have residual infected cells.

Not a fit: People without HIV or those whose virus has rare mutations that prevent CD4-mimetic binding are unlikely to benefit from this approach.

Why it matters

Potential benefit: If successful, these compounds could help shrink the reservoir of HIV-infected cells and make antibody-based treatments or prevention more effective.

How similar studies have performed: Related CD4-mimetic compounds have shown promising results in humanized mice and monkey models, but human use remains early-stage.

Where this research is happening

Boston, United States

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Acquired Immune Deficiency Syndrome VirusAcquired Immunodeficiency Syndrome Virus
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.