Blocking GPR171 to help immune cells fight cancer

The GPR171 pathway in cancer immunotherapy

NIH-funded research University of Colorado Denver · NIH-11306588

Researchers are looking at whether blocking a protein called GPR171 helps a patient’s immune cells attack tumors more effectively.

Quick facts

Grant typeR01 grant
Study typeNIH-funded research
Funding institutionUniversity of Colorado Denver NIH-funded
Lab location1 site (Aurora, UNITED STATES)
Project IDNIH-11306588 on NIH RePORTER

What this research studies

This project focuses on a pathway called BigLEN/GPR171 that appears to slow down the T cells that can kill cancer. The team studies T cells in the lab and uses mouse tumor models to see if drugs that block GPR171 boost antitumor immune responses. They will measure GPR171 protein levels after antigen stimulation, test GPR171 antagonists in tumors, and explore links between GPR171 and cannabinoid signaling. Findings could point toward new drugs or ways to improve current immunotherapies for patients.

Who could benefit from this research

Good fit: Patients with cancers treated by or resistant to immune checkpoint therapies (such as those receiving PD-1/CTLA-4–based treatments) would be the likely candidates for related future trials.

Not a fit: People with cancers that are unrelated to immune-driven tumor control or those ineligible for immunotherapy may not benefit from this approach.

Why it matters

Potential benefit: If successful, this work could lead to new treatments that make immune therapies work for more people and improve tumor control.

How similar studies have performed: Existing checkpoint drugs like PD-1 and CTLA-4 have proven benefit, and preliminary mouse studies reported here show blocking GPR171 can boost T cell antitumor activity, but GPR171 is a novel target without clinical trial evidence yet.

Where this research is happening

Aurora, UNITED STATES

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Conditions Cancer Patient
Last reviewed 2026-06-13 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.