A new oral treatment to prevent and reverse muscle loss in older adults

A Novel Small Molecule Oral Therapeutic to Prevent and Reverse Skeletal Muscle Atrophy in Aging Adults

NIH-funded research Ridgeline Therapeutics, LLC · NIH-10761425

This study is testing a new oral medication designed to help older adults keep their muscles strong and healthy, especially if they’ve been less active due to things like being in bed or not moving much.

Quick facts

Grant typeSbir 1 grant
Study typeNIH-funded research
Funding institutionRidgeline Therapeutics, LLC NIH-funded
Lab location1 site (Houston, UNITED STATES)
Project IDNIH-10761425 on NIH RePORTER

What this research studies

This research focuses on developing a small-molecule oral therapeutic aimed at preventing and reversing muscle atrophy in aging adults, particularly those who experience limited muscle use due to conditions like immobilization or bed rest. The approach involves inhibiting an enzyme called nicotinamide N-methyltransferase (NNMT), which plays a crucial role in cellular energy metabolism. By targeting this enzyme, the treatment aims to enhance muscle regeneration and repair, potentially improving strength and function in older adults. The clinical candidate, RT-002, is currently in preclinical studies, with plans for Phase 1 clinical trials starting soon.

Who could benefit from this research

Good fit: Ideal candidates for this research are older adults who are experiencing muscle atrophy due to disuse, such as those recovering from injuries or prolonged periods of inactivity.

Not a fit: Patients who are not experiencing muscle atrophy or those with muscle loss due to other underlying medical conditions may not benefit from this research.

Why it matters

Potential benefit: If successful, this research could provide a novel treatment option that helps aging adults maintain muscle mass and function, improving their overall health and independence.

How similar studies have performed: While there are ongoing developments in pharmaceutical interventions for muscle loss, this specific approach targeting NNMT is novel and has not been extensively tested in clinical settings.

Where this research is happening

Houston, UNITED STATES

Researchers

About this research

  1. This is an active NIH-funded research project — typically early-stage science, not a clinical trial accepting patient enrollment.
  2. Some NIH-funded labs run parallel clinical studies or seek volunteers for related work. To check, contact the principal investigator or institution listed above.
  3. For full project details, budget, and progress reports, visit the official NIH RePORTER page below.
Last reviewed 2026-06-10 by the Find a Trial editorial team. Information on this page is for educational purposes and is not medical advice. Always consult qualified healthcare professionals about clinical trial participation.